This information is for research and educational purposes only. No medical recommendations. Products are not approved for human use. For health questions, consult a doctor.

Lexicon

Regeneration

KPV Oral

The anti-inflammatory tripeptide KPV as a tablet, especially sensible for the gut because it is specifically taken up there.

1 min read 1 sources Titration Updated May 2026
Class
Anti-inflammatory tripeptide, oral
Use
Oral (tablet, 500mcg)
Focus
Gut, inflammation
Status
Preclinical (mainly gut models)

Getting started

Typical intake (research context)

Per-day figures. Oral KPV is especially obvious because it is taken up via the gut transporter PepT1.

Members only

Dosing recommendations are visible to logged-in members only. Logging in is free.

Log in / sign up

What is KPV Oral?

KPV Oral is the tablet form of the anti-inflammatory tripeptide KPV (see lexicon entry). With KPV especially, oral use is particularly obvious: the peptide is taken up via the gut transporter PepT1, which is even upregulated during inflammation.

How it works

KPV dampens central inflammation signaling routes directly inside cells. In the gut it is taken up via PepT1, so inflamed tissue absorbs KPV preferentially. That makes the oral form especially sensible for inflammatory gut topics.

The mechanism in detail is in the KPV entry.

How to take it

Oral, usually one tablet (500mcg) per day with some water.

Dosing

Members only

Dosing recommendations are visible to logged-in members only. Logging in is free.

Log in / sign up

What the research shows

A study (Dalmasso, 2008) showed that PepT1-mediated uptake of KPV markedly reduced inflammation in gut models, which is exactly what supports oral use. Large human studies are missing, KPV stays in the experimental range.

Side effects

  • Generally well tolerated.
  • Solid human data are limited.

Storage

Store dry, cool and protected from light, out of reach of children. Keep the original container closed and mind the expiry date.

Evidence

Sources

  1. 1 PepT1-mediated uptake of the tripeptide KPV reduces intestinal inflammation (preclinical). Dalmasso et al., Gastroenterology, 2008

Keep reading

More in the lexicon

In the shop

KPV Oral in the catalog

Sizes, prices and availability for research use. Straight from the lexicon to the product page.

View in shop